Molecule Details
InChIKeyHSOCYPPAQYZHMJ-UHFFFAOYSA-N
Compound Name1-[2-methoxy-4-[3-(trifluoromethyl)phenyl]phenyl]-2-oxo-N-pyrimidin-2-ylquinoline-6-sulfonamide
Canonical SMILESCOc1cc(-c2cccc(C(F)(F)F)c2)ccc1-n1c(=O)ccc2cc(S(=O)(=O)Nc3ncccn3)ccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.95
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15858 SCN9A Homo sapiens Human PF00520 PF24609 PF06512 PF11933 7.7 IC50 ChEMBL;BindingDB
Q9UQD0 SCN8A Homo sapiens Human PF00520 PF24609 PF06512 PF11933 6.2 IC50 ChEMBL;BindingDB