Molecule Details
InChIKeyHSMLVQPVLGLUCI-UHFFFAOYSA-N
Compound NameN2-(4-(benzo[d]thiazol-2-yl)-3-methoxyphenyl)-N4-(5-methyl-1H-pyrazol-3-yl)pyrimidine-2,4-diamine
Canonical SMILESCOc1cc(Nc2nccc(Nc3cc(C)[nH]n3)n2)ccc1-c1nc2ccccc2s1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.5
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 6.5 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 6.5 pIC50 TTD_MultiTarget