Molecule Details
InChIKeyHSEQWGUPLOFKEC-UHFFFAOYSA-N
Compound NameN-(3-Acetyl-6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-1-methyl-2-oxo-1,2-dihydro-1,8-naphthyridin-4-yl)methanesulfonamide
Canonical SMILESCC(=O)c1c(NS(C)(=O)=O)c2cc(-c3ccc(Cl)cc3)c(-c3ccc(Cl)cc3Cl)nc2n(C)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.09
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28335 HTR2C Homo sapiens Human PF00001 7.7 Ki ChEMBL
P21554 CNR1 Homo sapiens Human PF00001 7.5 IC50 ChEMBL
Q01959 SLC6A3 Homo sapiens Human PF00209 6.1 Ki ChEMBL