Molecule Details
InChIKeyHSBIXXNGKLUEIP-UHFFFAOYSA-N
Compound NameN-[3-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]acetamide
Canonical SMILESCC(=O)Nc1cccc(Nc2cc(NC3CC3)n3ncc(C#N)c3n2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P68400 CSNK2A1 Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
P19784 CSNK2A2 Homo sapiens Human PF00069 7.5 IC50 ChEMBL
P67870 CSNK2B Homo sapiens Human PF01214 7.2 IC50 ChEMBL