Molecule Details
InChIKeyHRVAZKKEGJGZOW-MOHJPFBDSA-N
Compound Name(5Z)-5-[4-[(7-chloro-2-oxochromen-4-yl)methylamino]phenyl]sulfonylimino-4-methyl-1,3,4-thiadiazole-2-sulfonamide
Canonical SMILESCn1nc(S(N)(=O)=O)s/c1=N\S(=O)(=O)c1ccc(NCc2cc(=O)oc3cc(Cl)ccc23)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL9.2
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 9.3 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 9.3 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 9.0 Ki ChEMBL;BindingDB