Molecule Details
InChIKeyHRKVZMGUPVYSKL-XTCLZLMSSA-N
Compound Name(NE)-N-[5-[1-(1-methylpiperidin-4-yl)-3-pyridin-4-ylpyrazol-4-yl]-2,3-dihydroinden-1-ylidene]hydroxylamine
Canonical SMILESCN1CCC(n2cc(-c3ccc4c(c3)CC/C4=N\O)c(-c3ccncc3)n2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.49
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P15056 BRAF Homo sapiens Human PF00130 PF07714 PF02196 9.5 IC50 ChEMBL;BindingDB
P27361 MAPK3 Homo sapiens Human PF00069 8.0 IC50 ChEMBL
P28482 MAPK1 Homo sapiens Human PF00069 8.0 IC50 ChEMBL