Molecule Details
InChIKeyHRFMJPIGMOWHLL-RUZDIDTESA-N
Compound Name1-[(R)-1-(4-Benzoyl-piperidine-1-carbonyl)-4-oxo-4-pyrrolidin-1-yl-butyl]-3-m-tolyl-urea
Canonical SMILESCc1cccc(NC(=O)N[C@H](CCC(=O)N2CCCC2)C(=O)N2CCC(C(=O)c3ccccc3)CC2)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.28
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P32238 CCKAR Homo sapiens Human PF00001 PF09193 7.3 pIC50 TTD_MultiTarget
P32239 CCKBR Homo sapiens Human PF00001 7.3 IC50 ChEMBL;BindingDB