Molecule Details
InChIKeyHRCUJSFALQORGR-UHFFFAOYSA-N
Compound Name4-[3-[4-Chloro-2-(3-methoxyphenyl)phenyl]-1-hydroxy-1-(3-methylimidazol-4-yl)prop-2-ynyl]benzonitrile
Canonical SMILESCOc1cccc(-c2cc(Cl)ccc2C#CC(O)(c2ccc(C#N)cc2)c2cncn2C)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.15
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 9.2 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 9.2 IC50 ChEMBL
P53609 PGGT1B Homo sapiens Human PF00432 6.1 IC50 ChEMBL;BindingDB