Molecule Details
InChIKeyHQXLJEBXFZNYOC-UHFFFAOYSA-N
Compound Name1-[3-Tert-butyl-1-(3-nitrophenyl)pyrazol-5-yl]-3-[3-(quinazolin-4-ylamino)phenyl]urea
Canonical SMILESCC(C)(C)c1cc(NC(=O)Nc2cccc(Nc3ncnc4ccccc34)c2)n(-c2cccc([N+](=O)[O-])c2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.79
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P00519 ABL1 Homo sapiens Human PF08919 PF07714 PF00017 PF00018 8.1 IC50 ChEMBL;BindingDB
P10721 KIT Homo sapiens Human PF00047 PF07714 7.5 IC50 ChEMBL