Molecule Details
InChIKeyHQWVFKGHUUEIMI-LBPRGKRZSA-N
Compound Name6-[(2S)-3-amino-2-hydroxypropyl]sulfonyl-3-[3-(2-amino-1H-imidazol-5-yl)phenyl]-2-(2H-tetrazol-5-yl)benzenesulfonamide
Canonical SMILESNC[C@H](O)CS(=O)(=O)c1ccc(-c2cccc(-c3c[nH]c(N)n3)c2)c(-c2nn[nH]n2)c1S(N)(=O)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.96
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.2 IC50 ChEMBL;BindingDB
Q9XAY4 blaVIM Pseudomonas aeruginosa Pathogen PF00753 8.9 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 8.7 IC50 BindingDB