Molecule Details
InChIKeyHQWSXGRKYMNJKY-OZXSUGGESA-N
Compound Name1-{2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinolin-3-ylmethyl}-3-phenyl-urea
Canonical SMILESCc1cc(O)cc(C)c1C[C@H](N)C(=O)N1Cc2ccccc2C[C@H]1CNC(=O)Nc1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41143 OPRD1 Homo sapiens Human PF00001 9.9 IC50 ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 9.0 IC50 ChEMBL;BindingDB
P41145 OPRK1 Homo sapiens Human PF00001 8.3 IC50 ChEMBL;BindingDB