Molecule Details
InChIKeyHQVRFXBZJOXOKH-NDBXHCKUSA-N
Canonical SMILESCCOC(=O)O[C@H](C)n1nnc(COC[C@H](C)N[C@H]2CC[C@H](Nc3cc(-c4cccc(NCC5(C#N)CCOCC5)n4)c(Cl)cn3)CC2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.43
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O60563 CCNT1 Homo sapiens Human PF00134 PF21797 8.4 IC50 ChEMBL;BindingDB
P50750 CDK9 Homo sapiens Human PF00069 8.4 IC50 ChEMBL