Molecule Details
InChIKeyHQRSMNLSFMUJPL-KOSHJBKYSA-N
Compound Name(2R)-N-(1-(6-aminopyridin-2-ylmethyl)piperidin-4-yl)-2-((1R)-3,3-difluorocyclopentyl)-2-hydroxy-2-phenylacetamide
Canonical SMILESNc1cccc(CN2CCC(NC(=O)[C@](O)(c3ccccc3)[C@@H]3CCC(F)(F)C3)CC2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.88
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11229 CHRM1 Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P20309 CHRM3 Homo sapiens Human PF00001 8.6 Ki ChEMBL;BindingDB
P08172 CHRM2 Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB