Molecule Details
InChIKeyHQKQOEMBHUHWCM-UHFFFAOYSA-N
Compound Name3-(2-(7-(Aminomethyl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl)quinolin-8-yloxy)-2,2-dimethylpropan-1-ol
Canonical SMILESCC(C)(CO)COc1cccc2ccc(-c3nnc4cc(CN)ccn34)nc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.46
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 9.2 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB