Molecule Details
InChIKeyHQIJOUHEHNIFNR-UHFFFAOYSA-N
Compound Name4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-naphthalen-2-yl)-1H-pyrrol-2-yl]-benzoic acid
Canonical SMILESCC1(C)CCC(C)(C)c2cc(-c3ccc(-c4ccc(C(=O)O)cc4)[nH]3)ccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.01
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P10276 RARA Homo sapiens Human PF00104 PF00105 9.3 IC50 ChEMBL;BindingDB
P13631 RARG Homo sapiens Human PF00104 PF00105 7.7 IC50 ChEMBL;BindingDB
P10826 RARB Homo sapiens Human PF00104 PF00105 7.0 IC50 ChEMBL;BindingDB