Molecule Details
InChIKeyHPVULTYLDIMYRI-RBKBAHBVSA-N
Compound Namecyclo[Arg-Cys(1)-Thr-His-D-Phe-Arg-N(Me)Trp-Pro-Ile-Cys(1)-Phe-Pro-Asp-Gly]
Canonical SMILESCC[C@H](C)[C@@H]1NC(=O)[C@@H]2CCCN2C(=O)[C@H](Cc2c[nH]c3ccccc23)N(C)C(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](Cc2cnc[nH]2)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@@H]2CSSC[C@H](NC1=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CC(=O)O)C(=O)NCC(=O)N[C@@H](CCCNC(=N)N)C(=O)N2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.16
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q01726 MC1R Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB
P32245 MC4R Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB
P33032 MC5R Homo sapiens Human PF00001 6.0 IC50 ChEMBL;BindingDB