Molecule Details
InChIKeyHOXJOAWSVADHMC-UHFFFAOYSA-N
Compound Name4-[1-(3-Carboxypropyl)-4-fluoro-2-methyl-7-[2-[4-[4-(2,3,4,6-tetrafluorophenyl)butoxy]phenyl]ethynyl]indol-3-yl]butanoic acid
Canonical SMILESCc1c(CCCC(=O)O)c2c(F)ccc(C#Cc3ccc(OCCCCc4c(F)cc(F)c(F)c4F)cc3)c2n1CCCC(=O)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.01
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y271 CYSLTR1 Homo sapiens Human PF00001 8.1 IC50 ChEMBL;BindingDB
Q9NS75 CYSLTR2 Homo sapiens Human PF00001 7.9 IC50 ChEMBL;BindingDB