Molecule Details
InChIKeyHOIIHACBCFLJET-NHCUHLMSSA-N
Compound Name1-(4-fluorophenyl)-4-((6bS,10aR)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3',4':4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)butan-1-one methylbenzenesulfonate
Canonical SMILESCN1CCN2c3c(cccc31)[C@H]1CN(CCCC(=O)c3ccc(F)cc3)CC[C@H]12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.3
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P28223 HTR2A Homo sapiens Human PF00001 8.3 Ki ChEMBL;BindingDB
P28335 HTR2C Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB