Molecule Details
InChIKeyHNQYRYXKHXZOGM-UHFFFAOYSA-N
Compound Name5-(5-Amino-2-[[3-(difluoromethoxy)pyridin-2-yl] methyl]-7-(1,3-oxazol-2-yl)-[1,2,4]triazolo[1,5-c] pyrimidin-8-yl)-l-methyl-1,2-dihydropyridin-2-one
Canonical SMILESCn1cc(-c2c(-c3ncco3)nc(N)n3nc(Cc4ncccc4OC(F)F)nc23)ccc1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.67
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30542 ADORA1 Homo sapiens Human PF00001 8.1 IC50 ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 8.0 IC50 ChEMBL;BindingDB
P29275 ADORA2B Homo sapiens Human PF00001 7.0 IC50 ChEMBL;BindingDB