Molecule Details
InChIKeyHNIKIMABKSIQOH-UHFFFAOYSA-N
Compound Name3-(4-amino-6-quinolyl)-2-(1H-tetrazol-5-yl)-6-(trifluoromethyl)benzenesulfonamide
Canonical SMILESNc1ccnc2ccc(-c3ccc(C(F)(F)F)c(S(N)(=O)=O)c3-c3nnn[nH]3)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.38
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q5GN09 vim-1 Klebsiella pneumoniae Pathogen PF00753 9.4 IC50 BindingDB
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 8.2 IC50 ChEMBL;BindingDB
P52699 Serratia marcescens Pathogen PF00753 7.5 IC50 BindingDB