Molecule Details
InChIKeyHMKRFXHMAJMWSE-LJFZDNNRSA-N
Canonical SMILESCc1cccc2c1NC(=O)[C@@H](NC(=O)[C@H](CCC(F)(F)F)[C@H](CC1CC(F)(F)C1)C(N)=O)N=C2c1cccc(F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.48
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q06330 RBPJ Homo sapiens Human PF09270 PF09271 PF20144 8.5 IC50 ChEMBL;BindingDB
P46531 NOTCH1 Homo sapiens Human PF00023 PF12796 PF00008 PF07645 PF12661 PF06816 PF07684 PF00066 8.5 IC50 ChEMBL;BindingDB