Molecule Details
InChIKeyHLPQICVVEMSECL-KRWDZBQOSA-N
Compound Name4-{5-[(S)-4-(3-Chloro-phenyl)-2-methyl-5-oxo-piperazin-1-ylmethyl]-imidazol-1-ylmethyl}-benzonitrile
Canonical SMILESC[C@H]1CN(c2cccc(Cl)c2)C(=O)CN1Cc1cncn1Cc1ccc(C#N)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.05
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.1 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.1 IC50 ChEMBL;BindingDB