Molecule Details
InChIKeyHLEHXKLGZMOEAM-UHFFFAOYSA-N
Compound Name3-(2-amino-4-fluoro-1,3-benzothiazol-6-yl)-2-(2H-tetrazol-5-yl)-6-(trifluoromethyl)benzenesulfonamide
Canonical SMILESNc1nc2c(F)cc(-c3ccc(C(F)(F)F)c(S(N)(=O)=O)c3-c3nnn[nH]3)cc2s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.42
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q5GN09 vim-1 Klebsiella pneumoniae Pathogen PF00753 9.8 IC50 BindingDB
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.4 IC50 ChEMBL;BindingDB
P52699 Serratia marcescens Pathogen PF00753 9.1 IC50 BindingDB