Molecule Details
InChIKeyHKYQMUOQXBQKOO-FXQIFTODSA-N
Compound Name[(2R,4S)-4-hydroxy-1-[(2S)-pyrrolidine-2-carbonyl]pyrrolidin-2-yl]boronic acid
Canonical SMILESO=C([C@@H]1CCCN1)N1C[C@@H](O)C[C@H]1B(O)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.37
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86TI2 DPP9 Homo sapiens Human PF19520 PF00930 PF00326 8.7 IC50 ChEMBL;BindingDB
Q6V1X1 DPP8 Homo sapiens Human PF19520 PF00930 PF00326 8.2 IC50 ChEMBL;BindingDB
P27487 DPP4 Homo sapiens Human PF00930 PF00326 8.2 IC50 ChEMBL;BindingDB