Molecule Details
InChIKeyHKSBXNVKPFTBIG-SHFRUIRLSA-N
Canonical SMILESCNc1nc(Nc2ccc(C(=O)N3CCN(C[C@H]4CC[C@H](CSC(C)(C)[C@H](NC(=O)C5(F)CC5)C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)CC4)CC3)cc2OC)ncc1Cl
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.76
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P40337 VHL Homo sapiens Human PF01847 PF17211 7.9 IC50 ChEMBL
Q5S007 LRRK2 Homo sapiens Human PF23745 PF23744 PF23748 PF16095 PF25497 PF13855 PF00069 PF08477 7.8 IC50 ChEMBL
Q96SW2 CRBN Homo sapiens Human PF02190 PF03226 7.6 IC50 ChEMBL