Molecule Details
InChIKeyHKOWUXNNUVZKQN-LBPRGKRZSA-N
Compound Name3,4-dichloro-2-(4-methoxy-3,3-dimethylbut-1-ynyl)-1-[(3S)-piperidin-3-yl]pyrrolo[2,3-b]pyridine-6-carboxamide
Canonical SMILESCOCC(C)(C)C#Cc1c(Cl)c2c(Cl)cc(C(N)=O)nc2n1[C@H]1CCCNC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.72
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q12809 KCNH2 Homo sapiens Human PF00027 PF00520 PF13426 9.0 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 8.8 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB