Molecule Details
InChIKeyHKGUHEGKBLYKHY-QMOZSOIISA-N
Compound NameAzd-3409
Canonical SMILESCSCC[C@H](NC(=O)c1cc(NC[C@@H]2C[C@H](SC(=O)c3cccnc3)CN2)ccc1CCc1ccc(F)cc1)C(=O)OC(C)C
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.7
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 9.0 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 9.0 Ki ChEMBL;BindingDB
P53609 PGGT1B Homo sapiens Human PF00432 8.1 Ki ChEMBL