Molecule Details
InChIKeyHKDOASHONDCKDU-UHFFFAOYSA-N
Compound Name2-[4-[4-(5-Chloro-2-pyridinyl)piperazin-1-yl]butyl]-1,3-benzothiazole
Canonical SMILESClc1ccc(N2CCN(CCCCc3nc4ccccc4s3)CC2)nc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.12
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21917 DRD4 Homo sapiens Human PF00001 8.3 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB