Molecule Details
InChIKeyHJUDFJRTVGXBRF-UHFFFAOYSA-N
Compound NameN-[4-Methyl-3-(1h-1,2,4-Triazol-5-Yl)thiophen-2-Yl]-2-(2-Oxo-3,4-Dihydroquinolin-1(2h)-Yl)acetamide
Canonical SMILESCc1csc(NC(=O)CN2C(=O)CCc3ccccc32)c1-c1ncn[nH]1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.54
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P53779 MAPK10 Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB