Molecule Details
InChIKeyHIWTYESDVJEVCS-UHFFFAOYSA-N
Compound Name3-Methyl-5-[1-(6-piperazin-1-yl-2-pyridinyl)pyrazolo[4,3-c]pyridin-6-yl]-1,2-thiazole
Canonical SMILESCc1cc(-c2cc3c(cn2)cnn3-c2cccc(N3CCNCC3)n2)sn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.98
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 9.5 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 9.4 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.1 Ki ChEMBL;BindingDB