Molecule Details
InChIKeyHIQIMBYLAJXNOK-UHFFFAOYSA-N
Compound Name4-(5-Methyl-1H-pyrazol-3-ylamino)-2-(4-nitrobenzyl)-2Hphthalazin-1-one
Canonical SMILESCc1cc(Nc2nn(Cc3ccc([N+](=O)[O-])cc3)c(=O)c3ccccc23)n[nH]1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.65
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 7.0 pIC50 TTD_MultiTarget
Q96GD4 AURKB Homo sapiens Human PF00069 6.0 IC50 ChEMBL;BindingDB