Molecule Details
InChIKeyHIASHEATKNRFJC-UHFFFAOYSA-N
Compound Name6-(2-Morpholinoethylamino)-4-(4-(phenylthio)phenylamino)-1,7-naphthyridine-3-carbonitrile
Canonical SMILESN#Cc1cnc2cnc(NCCN3CCOCC3)cc2c1Nc1ccc(Sc2ccccc2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.12
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P41279 MAP3K8 Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
Q02750 MAP2K1 Homo sapiens Human PF00069 6.0 IC50 ChEMBL;BindingDB