Molecule Details
InChIKeyHHYOQRDAWFAMAJ-INIZCTEOSA-N
Compound Name(S)-3-(6-bromo-4-methyl-1H-benzo[d]imidazol-2-yl)-4-(1-hydroxy-3-phenylpropan-2-ylamino)pyridin-2(1H)-one
Canonical SMILESCc1cc(Br)cc2[nH]c(-c3c(N[C@H](CO)Cc4ccccc4)cc[nH]c3=O)nc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.64
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P05177 CYP1A2 Homo sapiens Human PF00067 7.3 IC50 ChEMBL;BindingDB
P33261 CYP2C19 Homo sapiens Human PF00067 6.5 IC50 ChEMBL
P11712 CYP2C9 Homo sapiens Human PF00067 6.1 IC50 ChEMBL;BindingDB