Molecule Details
InChIKeyHHIRKUWNXWZRBC-MHZLTWQESA-N
Compound NameN-[(1S)-1-[5-(2-methoxy-3-quinolyl)-1H-imidazol-2-yl]-7-oxo-nonyl]-2-methyl-2-azaspiro[3.5]nonane-7-carboxamide
Canonical SMILESCCC(=O)CCCCC[C@H](NC(=O)C1CCC2(CC1)CN(C)C2)c1ncc(-c2cc3ccccc3nc2OC)[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.87
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O15379 HDAC3 Homo sapiens Human PF00850 8.8 IC50 ChEMBL;BindingDB
Q92769 HDAC2 Homo sapiens Human PF00850 8.4 IC50 ChEMBL;BindingDB
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 6.3 IC50 ChEMBL;BindingDB