Molecule Details
InChIKeyHHHGGOMKUAYOJZ-HHHXNRCGSA-N
Compound Name3-Amino-N-((R)-1-(2,4-dichloro-benzyl)-2-oxo-2-{4-[1-(phenylacetylamino-methyl)-cyclohexyl]-piperazin-1-yl}-ethyl)-propionamide
Canonical SMILESNCCC(=O)N[C@H](Cc1ccc(Cl)cc1Cl)C(=O)N1CCN(C2(CNC(=O)Cc3ccccc3)CCCCC2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.77
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P32245 MC4R Homo sapiens Human PF00001 8.1 Ki ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB
P33032 MC5R Homo sapiens Human PF00001 6.0 Ki ChEMBL;BindingDB