Molecule Details
InChIKeyHHCRCIWZXNRZMQ-UHFFFAOYSA-N
Compound NameN-[(4-chlorophenyl)methyl]-2-(5-fluoro-2,4-dioxopyrimidin-1-yl)-N-[2-(4-sulfamoylphenyl)ethyl]acetamide
Canonical SMILESNS(=O)(=O)c1ccc(CCN(Cc2ccc(Cl)cc2)C(=O)Cn2cc(F)c(=O)[nH]c2=O)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.02
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16790 CA9 Homo sapiens Human PF00194 8.4 Ki ChEMBL;BindingDB
O43570 CA12 Homo sapiens Human PF00194 8.2 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 7.5 Ki ChEMBL;BindingDB