Molecule Details
InChIKeyHGSQEWOPIVMPGD-VIFPVBQESA-N
Compound Name3-[(3S)-3-aminopiperidin-1-yl]-6-(azetidin-3-ylsulfonyl)-2-(2H-tetrazol-5-yl)benzenesulfonamide
Canonical SMILESN[C@H]1CCCN(c2ccc(S(=O)(=O)C3CNC3)c(S(N)(=O)=O)c2-c2nnn[nH]2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.24
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q5GN09 vim-1 Klebsiella pneumoniae Pathogen PF00753 8.0 IC50 BindingDB
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 7.1 IC50 ChEMBL;BindingDB
Q79MP6 blaIMP-1 Pseudomonas aeruginosa Pathogen PF00753 6.6 IC50 ChEMBL;BindingDB