Molecule Details
InChIKeyHGRGBTOFFWBXHE-UHFFFAOYSA-N
Compound Name3-amino-6-(2-fluorophenyl)-N-(4-pyridin-4-yl-3-pyridinyl)pyridine-2-carboxamide
Canonical SMILESNc1ccc(-c2ccccc2F)nc1C(=O)Nc1cnccc1-c1ccncc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.43
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 8.1 Ki ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 7.7 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.5 Ki ChEMBL;BindingDB