Molecule Details
InChIKeyHGOSXKUMUKYUKG-UHFFFAOYSA-N
Compound Name4-cyano-N-(2-cyclohexenyl-4-(pyridin-4-yl)phenyl)-1H-imidazole-2-carboxamide
Canonical SMILESN#Cc1c[nH]c(C(=O)Nc2ccc(-c3ccncc3)cc2C2=CCCCC2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.98
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11712 CYP2C9 Homo sapiens Human PF00067 8.5 IC50 ChEMBL;BindingDB
P07333 CSF1R Homo sapiens Human PF00047 PF25305 PF07714 8.3 IC50 ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 7.1 IC50 ChEMBL;BindingDB