Molecule Details
InChIKeyHFSFBCFFSSYGFK-UHFFFAOYSA-N
Compound Name1-[4-[1-ethyl-4-[2-[3-(morpholin-4-ylmethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl]pyrazol-3-yl]phenyl]-3-phenylurea
Canonical SMILESCCn1cc(-c2ccnc3[nH]c(-c4cccc(CN5CCOCC5)c4)cc23)c(-c2ccc(NC(=O)Nc3ccccc3)cc2)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.1
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 7.2 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 7.0 pIC50 TTD_MultiTarget