Molecule Details
InChIKeyHFOKVVVCWLIUBP-UHFFFAOYSA-N
Compound Name5-{1-[(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-4-fluoro-2,3-dihydro-1H-indol-5-yl}-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
Canonical SMILESCc1cc(C)n(CC(=O)N2CCc3c2ccc(-c2cn(C)c4ncnc(N)c24)c3F)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.42
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9NZJ5 EIF2AK3 Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
Q9BQI3 EIF2AK1 Homo sapiens Human PF22949 PF00069 7.2 IC50 ChEMBL;BindingDB
P19525 EIF2AK2 Homo sapiens Human PF00035 PF00069 7.0 IC50 ChEMBL;BindingDB