Molecule Details
InChIKeyHFBOFILREKLDAP-UHFFFAOYSA-N
Compound Name2,3,5,6-Tetrafluoro-N-{4-[2-(4-sulfamoyl-phenyl)-ethylsulfamoyl]-phenyl}-benzamide
Canonical SMILESNS(=O)(=O)c1ccc(CCNS(=O)(=O)c2ccc(NC(=O)c3c(F)c(F)cc(F)c3F)cc2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.97
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16790 CA9 Homo sapiens Human PF00194 8.1 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 7.9 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 7.9 pIC50 TTD_MultiTarget