Molecule Details
InChIKeyHEZDUVOOOSBRGR-LOACHALJSA-N
Compound Name(3S)-7-[3-(2,2-dimethyl-1,3-dithiolan-4-yl)propanoylamino]-3,4-dihydro-1H-isochromene-3-carboxylic acid
Canonical SMILESCC1(C)SCC(CCC(=O)Nc2ccc3c(c2)CO[C@H](C(=O)O)C3)S1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.39
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P18031 PTPN1 Homo sapiens Human PF00102 6.5 IC50 ChEMBL;BindingDB
P17706 PTPN2 Homo sapiens Human PF00102 6.4 IC50 ChEMBL;BindingDB
P10586 PTPRF Homo sapiens Human PF00041 PF07679 PF00102 6.3 IC50 ChEMBL;BindingDB