Molecule Details
InChIKeyHEOZBPOPPDUPGK-UHFFFAOYSA-N
Compound Name8-Cyclopropyl-2-[(4-methylpiperazin-1-yl)methyl][1]benzofuro[3,2-d]pyrimidin-4(3H)-one
Canonical SMILESCN1CCN(Cc2nc3c(oc4ccc(C5CC5)cc43)c(=O)[nH]2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.37
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.1 IC50 ChEMBL;BindingDB