Molecule Details
InChIKeyHENCYENWBZRSLR-UHFFFAOYSA-N
Compound NameN-isopropyl-4-(3-(1-(methylsulfonyl)piperidin-4-yl)-1H-pyrazol-4-yl)pyrimidin-2-amine
Canonical SMILESCC(C)Nc1nccc(-c2c[nH]nc2C2CCN(S(C)(=O)=O)CC2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.77
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 7.0 Ki ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 6.7 IC50 ChEMBL
P53779 MAPK10 Homo sapiens Human PF00069 6.7 IC50 ChEMBL