Molecule Details
InChIKeyHEJWDMSZDBYDME-UHFFFAOYSA-N
Compound NameUS11111247, Example 36
Canonical SMILESCN1CCN(c2ncc3[nH]nc(-c4cnn(C)c4)c3n2)CC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.36
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21802 FGFR2 Homo sapiens Human PF07679 PF13927 PF07714 6.5 IC50 ChEMBL;BindingDB
P22607 FGFR3 Homo sapiens Human PF21165 PF07679 PF13927 PF07714 6.5 IC50 ChEMBL;BindingDB
P11362 FGFR1 Homo sapiens Human PF07679 PF00047 PF07714 6.0 IC50 ChEMBL