Molecule Details
InChIKeyHDECOLDRAJGUTB-UHFFFAOYSA-N
Compound Name2-(2,6-Difluorophenyl)-4-(4-piperazin-1-ylquinolin-6-yl)-1,3-thiazole
Canonical SMILESFc1cccc(F)c1-c1nc(-c2ccc3nccc(N4CCNCC4)c3c2)cs1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 8.3 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.7 IC50 ChEMBL;BindingDB