Molecule Details
InChIKeyHCSMZVMWZMSHSC-LZNHGOJSSA-N
Canonical SMILESCC1=C(C(=O)N[C@H](C)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CC2CCCCC2)C(=O)[C@@]2(C)CO2)Cc2ccccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.58
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P28074 PSMB5 Homo sapiens Human PF00227 7.8 IC50 ChEMBL;BindingDB
P28062 PSMB8 Homo sapiens Human PF00227 7.4 IC50 ChEMBL;BindingDB