Molecule Details
InChIKeyHCDXOVUMIOIELK-UHFFFAOYSA-N
Compound Name[4-[[7-Cyclopentyl-6-(1,5-dimethylpyrazol-4-yl)pyrrolo[2,3-d]pyrimidin-2-yl]amino]-1-methylpyrrol-2-yl]-(4-methylpiperazin-1-yl)methanone
Canonical SMILESCc1c(-c2cc3cnc(Nc4cc(C(=O)N5CCN(C)CC5)n(C)c4)nc3n2C2CCCC2)cnn1C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.86
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 8.7 IC50 ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
P06493 CDK1 Homo sapiens Human PF00069 6.5 IC50 ChEMBL;BindingDB