Molecule Details
InChIKeyHBGMCCARHCLDCH-AREUJWMLSA-N
Canonical SMILESCOc1cc(C(=O)N[C@H]2C(O)O[C@H](CNS(=O)(=O)c3cccc(Cl)c3Cl)[C@@H](O)[C@@H]2O)cc(-c2ccc(C#N)cc2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.85
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P19367 HK1 Homo sapiens Human PF00349 PF03727 8.1 IC50 ChEMBL;BindingDB
P52789 HK2 Homo sapiens Human PF00349 PF03727 7.6 IC50 ChEMBL;BindingDB